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Convergent catalytic asymmetric synthesis of camptothecin analog GI147211C  • ARTICLE Francis G. Fang, Donald D. Bankston, Edward M. Huie, M. Ross Johnson, Myung-Chol Kang, Craig S. LeHoullier, George C. Lewis, Thomas C. Lovelace, Melissa W. Lowery, Darryl L. McDougald et al. Abstract | Abstract + References | PDF (977 K) |
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Double stereodifferentiation in the Lewis acid promoted C-glycosidation of activated glycals with chiral (E)-crotylsilanes  • ARTICLE James S. Panek and Jennifer V. Schaus Abstract | Abstract + References | PDF (652 K) |
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Synthesis of the orally active spiroindoline-based growth hormone secretagogue, MK-677  • ARTICLE Peter E. Maligres, Ioannis Houpis, Kai Rossen, Audrey Molina, Jess Sager, Veena Upadhyay, Kenneth M. Wells, Robert A. Reamer, Joseph E. Lynch, David Askin et al. Abstract | Abstract + References | PDF (705 K) |
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Synthesis of : Sugar moiety of antitumor antibiotic bleomycin  • ARTICLE Tetsuta Oshitari, Masakatsu Shibasaki, Takeshi Yoshizawa, Masahiro Tomita, Ken-ichi Takao and Susumu Kobayashi Abstract | Abstract + References | PDF (892 K) |
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The 14C radiolabelled synthesis of the cholesterol absorption inhibitor CP-148,623. A novel method for the incorporation of a 14C label in enones  • ARTICLE Michael P. DeNinno and Keith E. McCarthy Abstract | Abstract + References | PDF (612 K) |
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Synthesis of the novel mannosidase inhibitors (3R)- and (3S)-3-(hydroxymethyl)swainsonine  • ARTICLE Erik J. Hembre and William H. Pearson Abstract | Abstract + References | PDF (804 K) |
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Synthesis of bis-abasic cyclic dinucleotide, bis-(3→5)-cyclic Bis(1,4-anhydro-2-deoxy--erythro-pentitol-3-phosphate), an inhibitor HIV-1 integrase  • ARTICLE H. Keith Chenault and Robert F. Mandes Abstract | Abstract + References | PDF (391 K) |
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Ring opening of sialyllactones with glycine esters: Synthesis of selectively protected glycinyl-NeuAc saccharopeptides  • ARTICLE Jacquelyn Gervay, P. S. Ramamoorthy and Nellie N. Mamuya Abstract | Abstract + References | PDF (491 K) |
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Practical total synthesis of (+)-Camptothecin: The full story  • ARTICLE Marco A. Ciufolini and Frank Roschangar Abstract | Abstract + References | PDF (889 K) |
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Synthesis of pyranose glycals via tungsten and molybdenum pentacarbonyl-induced alkynol cyclizations  • ARTICLE Frank E. McDonald and Hugh Y. H. Zhu Abstract | Abstract + References | PDF (500 K) |
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Transformation of 1-(1,2-propadienyl)cyclopropanols into substituted hydroquinones employing octacarbonyldicobalt  • ARTICLE Yufu Owada, Takeshi Matsuo and Nobuharu Iwasawa Abstract | Abstract + References | PDF (975 K) |
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Total synthesis of (+)-curacin A, a marine cytotoxic agent  • ARTICLE Michael Z. Hoemann, Konstantinos A. Agrios and Jeffrey Aubé Abstract | Abstract + References | PDF (865 K) |
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Application of the oxa-di--methane photoisomerization in the rearrangement of carbocycles possessing bridgehead unsaturation  • ARTICLE R. Michael Corbett, Chee-Seng Lee, Michelle M. Sulikowski, Joseph Reibenspies and Gary A. Sulikowski Abstract | Abstract + References | PDF (596 K) |
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Synthesis of CMP-sialic acid conjugates: Substrates for the enzymatic synthesis of natural and designed sialyl oligosaccharides  • ARTICLE Mark D. Chappell and Randall L. Halcomb Abstract | Abstract + References | PDF (693 K) |
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Tandem Michael addition and azanorbornane substance-P antagonists  • ARTICLE B. T. O'Neill, P. F. Thadeio, M. W. Bundesmann, A. M. Elder, S. McLean and D. K. Bryce Abstract | Abstract + References | PDF (1310 K) |
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Enantioselective synthesis of -amino acids from glycine t-butyl ester  • ARTICLE Tsai-Lung Yeh, Chun-Chen Liao and Biing-Jiun Uang Abstract | Abstract + References | PDF (655 K) |
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A convergent synthesis of (+)-pancratistatin based on intramolecular electrophilic aromatic substitution  • ARTICLE Timothy J. Doyle, Martin Hendrix, Donald VanDerveer, Sahar Javanmard and John Haseltine Abstract | Abstract + References | PDF (1252 K) |
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A facile solution and solid phase synthesis of phosphotyrosine mimetic -4-[diethylphosphono(difluoromethyl)]-phenylalanine (F2Pmp(EtO)2) derivatives  • ARTICLE Maher N. Qabar, Jan Urban and Michael Kahn Abstract | Abstract + References | PDF (407 K) |
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The kinetics and thermodynamics of bicyclic ketal formation: An application to the synthesis of the zaragozic acids  • ARTICLE Sayee G. Hegde and David C. Myles Abstract | Abstract + References | PDF (652 K) |
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6-Thio-2′-deoxyinosine: Synthesis, incorporation, and evaluation as a postsynthetically modifiable base in oligonucleotides  • ARTICLE Robert S. Coleman, John C. Arthur and Jason L. McCary Abstract | Abstract + References | PDF (621 K) |
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An enantioselective route to trans-2,6-disubstituted piperidines  • ARTICLE Samuel Chackalamannil and Yuguang Wang Abstract | Abstract + References | PDF (389 K) |
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A titanium (IV) mediated one-pot double condensation synthesis of 5,6-dihydro-4H-pyran-4-ones  • ARTICLE Joel Morris, Donn G. Wishka, George P. Luke, Thomas M. Judge and Ronald B. Gammill Abstract | Abstract + References | PDF (584 K) |
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Asymmetric Michael addition of nitroalkanes to prochiral acceptors catalyzed by proline rubidium salts  • ARTICLE Masahiko Yamaguchi, Yoshihiro Igarashi, Ravinder S. Reddy, Tai Shiraishi and Masahiro Hirama Abstract | Abstract + References | PDF (896 K) |
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Preface  • EDITORIAL Samuel J. Danishefsky Abstract | Abstract + References | PDF (55 K) |
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Contributors to this issue  • MISCELLANEOUS PDF (38 K) |
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Graphical abstracts  • ABSTRACT PDF (297 K) |
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